Abstract
The present application relates to a process for the preparation of 2-{3-[4-(1H-indazol-5-ylamino)-2-quinazolinyl]phenoxy}-N-(propan-2-yl) acetamide represented by the following structural formula-1, which is referred to as Belumosudil and its intermediate preparation thereof.
Formula-1.
The present application also relates to novel crystalline forms of Belumosudil, its mesylate and its intermediate and preparation thereof.
Creative Commons License
This work is licensed under a Creative Commons Attribution 4.0 License.
Recommended Citation
MSN Laboratories Private Limited, R&D Center; Srinivasan Thirumalai Rajan; Sajja Eswaraiah; Sagyam Rajeshwar Reddy; Keshavareddy Navin Kumar Reddy; Kootikanti Krishnaiah; Yata Murali and Utnoori Venkata Chary, "A process for the preparation of 2-{3-[4-(1H-indazol-5-ylamino)-2-quinazolinyl] phenoxy}-N-(propan-2-yl) acetamide and its salts", Technical Disclosure Commons, (November 01, 2023)
https://www.tdcommons.org/dpubs_series/6378