A PROCESS FOR THE PREPARATION OF (4-CHLORO-7-(2-((S)-1-(2- ((3BS,4AR)-5,5-DIFLUORO-3-(TRIFLUOROMETHYL)-3B,4,4A,5-TETRAHYDRO-1HCYCLOPROPA[3,4]CYCLOPENTA[1,2-C]PYRAZOL-1-YL)ACETAMIDO)-2-(3,5-DIFLUOROPHENYL)ETHYL)-6-(3-METHYL-3-(METHYLSULFONYL) BUT-1-YN-1-YL)PYRIDIN-3-YL)-1-(2,2,2-TRIFLUOROETHYL)-1H-INDAZOL3-YL)(METHYLSULFONYL)AMIDE SODIUM

Inventor(s)

• Lee Pharma Limited

Abstract

The present disclosure relates to (4-chloro-7-(2-((S)-1-(2-((3bS,4aR)-5,5-difluoro-3-(trifluoromethyl)-3b,4,4a,5-tetrahydro-1Hcyclopropa[3,4]cyclopenta[1,2-c]pyrazol-1-yl) acetamido)-2-(3,5-difluorophenyl)ethyl)-6-(3-methyl-3-(methylsulfonyl)but-1-yn-1-yl) pyridin-3-yl)-1-(2,2,2-trifluoroethyl)-1H-indazol3-yl)(methylsulfonyl)amide Sodium, is represented by following structural formula (1) and its process for the preparation thereof.

Creative Commons License

This work is licensed under a Creative Commons Attribution 4.0 License.

Recommended Citation

Lee Pharma Limited, "A PROCESS FOR THE PREPARATION OF (4-CHLORO-7-(2-((S)-1-(2- ((3BS,4AR)-5,5-DIFLUORO-3-(TRIFLUOROMETHYL)-3B,4,4A,5-TETRAHYDRO-1HCYCLOPROPA[3,4]CYCLOPENTA[1,2-C]PYRAZOL-1-YL)ACETAMIDO)-2-(3,5-DIFLUOROPHENYL)ETHYL)-6-(3-METHYL-3-(METHYLSULFONYL) BUT-1-YN-1-YL)PYRIDIN-3-YL)-1-(2,2,2-TRIFLUOROETHYL)-1H-INDAZOL3-YL)(METHYLSULFONYL)AMIDE SODIUM", Technical Disclosure Commons, (July 20, 2026)
https://www.tdcommons.org/dpubs_series/11056